prof. dr. A.S.S. (Alexander) Dömling

Professor and chair Drug Design Group

prof. dr. A.S.S. (Alexander) Dömling
Telephone:
E-mail:
a.s.s.domling rug.nl

Research

Postal address:
A Deusinglaan1
Gebouw 3211, ruimte 0470
9713 AV
Groningen
Netherlands
Phone: +31 50 363 3307Fax: +31 50 363 6908
  1. 2020
  2. van der Vlag, R., Unver, M. Y., Felicetti, T., Twarda-Clapa, A., Kassim, F., Ermis, C., ... Hirsch, A. K. H. (2020). Optimized Inhibitors of MDM2 via an Attempted Protein-Templated Reductive Amination. ChemMedChem, 15(4), 370-375. https://doi.org/10.1002/cmdc.201900574
  3. Abdelraheem, E. M. M., Goodwin, I., Shaabani, S., de Haan, M. P., Kurpiewska, K., Kalinowska-Tłuścik, J., & Dömling, A. (2020). 'Atypical Ugi' tetrazoles. Chemical communications (Cambridge, England), 56(12), 1799-1802. https://doi.org/10.1039/c9cc09194g
  4. 2019
  5. Neochoritis, C. G., Zarganes-Tzitzikas, T., Novotna, M., Mitrikova, T., Wang, Z., Kurpiewska, K., ... Domling, A. (2019). Isocyanide-Based Multicomponent Reactions of Free Phenylboronic Acids. European Journal of Organic Chemistry, 2019(35), 6132-6137. https://doi.org/10.1002/ejoc.201901187
  6. Batista, F. A., Bosch, S. S., Butzloff, S., Lunev, S., Meissner, K. A., Linzke, M., ... Wrenger, C. (2019). Oligomeric protein interference validates druggability of aspartate interconversion in Plasmodium falciparum. MicrobiologyOpen, 8(7), [e779]. https://doi.org/10.1002/mbo3.779
  7. Ghonchepour, E., Neochoritis, C. G., Kurpiewska, K., Kalinowska-Tluscik, J., Islami, M. R., & Domling, A. (2019). Glycoconjugates via Phosphorus Ylides. European Journal of Organic Chemistry, 2019(22), 3632-3635. https://doi.org/10.1002/ejoc.201900434
  8. Skalniak, L., Twarda-Clapa, A., Neochoritis, C. G., Surmiak, E., Machula, M., Wisniewska, A., ... Holak, T. A. (2019). A fluorinated indole-based MDM2 antagonist selectively inhibits the growth of p53wt osteosarcoma cells. The FEBS Journal, 286(7), 1360-1374. https://doi.org/10.1111/febs.14774
  9. Neochoritis, C. G., Kazemi Miraki, M., Abdelraheem, E. M. M., Surmiak, E., Zarganes-Tzitzikas, T., Łabuzek, B., ... Dömling, A. (2019). Design of indole- and MCR-based macrocycles as p53-MDM2 antagonists. Beilstein Journal of Organic Chemistry, 15, 513-520. https://doi.org/10.3762/bjoc.15.45
  10. 2018
  11. dos Santos Clemente, G., Zarganes Tzitzikas, T., F. Antunes, I., Elsinga, P. H., & Dömling, A. (2018). MCR scaffolds as synthons for the development of PET radiotracers. 95. Abstract from 7th International Conference on
    Multicomponent Reactions and Related Chemistry, Düsseldorf, Germany.
  12. Doemling, A., Abdelraheem, E. M. M., Rudrakshula, M., Khalesi, M., Neochoritis, C., Patil, P., & Shaabani, S. (2018). Very short and diverse synthesis of artificial marcocycles. Abstracts of Papers of the American Chemical Society, 256.
Previous 1 2 3 4 5 6 Next

ID: 413873