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How to find us prof. dr. A.S.S. (Alexander) Dömling

prof. dr. A.S.S. (Alexander) Dömling

Professor and chair Drug Design Group

prof. dr. A.S.S. (Alexander) Dömling

Faculty of Science and Engineering

Telephone:

+31 50 36 33307

+31 50 36 33336 (secretariat)

+31 50 36 37582 (fax)

E-mail:

a.s.s.domling rug.nl

Homepage ORCID Research Portal

Publications

Enabling large-scale design, synthesis and validation of small molecule protein-protein antagonists

Koes, D., Khoury, K., Huang, Y., Wang, W., Bista, M., Popowicz, G. M., Wolf, S., Holak, T. A., Dömling, A. & Camacho, C. J., 12-Mar-2012 , In: PLoS ONE. 7 , 3 , 8 p. , e32839.

Research output: Contribution to journal › Article › Academic › peer-review

Chemistry and Biology Of Multicomponent Reactions

Domling, A. , Wang, W. & Wang, K., Jun-2012 , In: Chemical reviews. 112 , 6 , p. 3083-3135 53 p.

Research output: Contribution to journal › Review article › peer-review

Efficient Assembly of Iminodicarboxamides by a "Truly" Four-Component Reaction

Khoury, K., Sinha, M. K., Nagashima, T., Herdtweck, E. & Domling, A. , 2012 , In: Angewandte Chemie-International Edition. 51 , 41 , p. 10280-10283 4 p.

Research output: Contribution to journal › Article › Academic › peer-review

Correction to "Benchmark of Generic Shapes for Macrocycles"

Reyes Romero, A. , Ruiz-Moreno, A. J., Groves, M. R. , Velasco-Velázquez, M. & Dömling, A. , 25-May-2021 , (E-pub ahead of print) In: Journal of chemical information and modeling.

Research output: Contribution to journal › Article › Academic › peer-review

Design, Synthesis, and Biological Evaluation of Imidazopyridines as PD-1/PD-L1 Antagonists

Butera, R. , Ważyńska, M. , Magiera-Mularz, K., Plewka, J., Musielak, B., Surmiak, E., Sala, D., Kitel, R., de Bruyn, M. , Nijman, H. W. , Elsinga, P. H. , Holak, T. A. & Dömling, A. , 2021 , In: Bioorganic & Medicinal Chemistry Letters. 12 , 5 , p. 768-773 6 p.

Research output: Contribution to journal › Article › Academic › peer-review

In Silico Design and Selection of New Tetrahydroisoquinoline-Based CD44 Antagonist Candidates

Ruiz-Moreno, A. J., Reyes-Romero, A. , Dömling, A. & Velasco-Velázquez, M. A., 2021 , In: Molecules. 26 , 7 , 17 p. , 1877.

Research output: Contribution to journal › Article › Academic › peer-review

Mapping arginase expression with 18F-fluorinated late-generation arginase inhibitors derived from quaternary α-amino acids

Clemente, G. S. , F Antunes, I. , Kurhade, S., Berg, M. V. D. , Sijbesma, J. W. A., Waarde, A. V. , Buijsmam, R. C., Willemsen-Seegers, N., Gosens, R. , Meurs, H. , Dömling, A. & Elsinga, P. H. , 1-Mar-2021 , In: Journal of Nuclear Medicine. 62 , 3

Research output: Contribution to journal › Article › Academic › peer-review

Marriage of high throughput synthesis and high throughput protein crystallography

Doemling, A. , Sutanto, F. , Shaabani, S. , Oerlemans, R. , Deniz, E., Patil, P. , Hadian, M., Wang, M., Sharpe, M. E. & Groves, M. R. , 7-Jun-2021 , (E-pub ahead of print) In: Angewandte Chemie (International ed. in English).

Research output: Contribution to journal › Article › Academic › peer-review

Multicomponent reaction-derived covalent inhibitor space

Sutanto, F. , Shaabani, S. , Neochoritis, C. G., Zarganes-Tzitzikas, T., Patil, P., Ghonchepour, E. & Dömling, A. , Feb-2021 , In: Science Advances. 7 , 6 , 11 p. , 9307.

Research output: Contribution to journal › Article › Academic › peer-review

Nanoscale, automated, high throughput synthesis and screening for the accelerated discovery of protein modifiers

Gao, K. , Shaabani, S. , Xu, R. , Zarganes-Tzitzikas, T., Gao, L. , Ahmadianmoghaddam, M. , Groves, M. R. & Domling, A. , May-2021 , In: RSC Medicinal Chemistry. 12 , 5 , p. 809-818 10 p.

Research output: Contribution to journal › Article › Academic › peer-review

All (326) publications

Press/media

Automated and Accelerated Synthesis of Indole Derivatives on a Nano-Scale

Alex Dömling

29/08/2019

Press/Media: Research › Academic

Computational chemistry, Medicijnen & Farmacologie, Organische chemie

Alex Dömling

26/07/2019

Press/Media: Research › Academic

Supersnelle boorzuurchemie dankzij syntheserobot

Alex Dömling

26/07/2019

Press/Media: Research › Academic

Supersnelle boorzuurchemie dankzij syntheserobot

Alex Dömling

26/07/2019

Press/Media: Research › Academic

Snelle methode voor synthese van kandidaat-geneesmiddelen. High-throughput systeem levert mogelijk middel tegen tuberculose op

Alex Dömling

09/07/2019

Press/Media: Research › Academic

Small-volume, high-throughput organic synthesis. New method synthesizes and evaluates large number of drug leads

Alex Dömling

09/07/2019

Press/Media: Research › Academic

Acoustic robot races through chemical reactions

Alexander Dömling

11/03/2019

Press/Media: Research › Professional

Acoustic robot races through chemical reactions. Using ultrasound to dispense reagents could accelerate the development of synthetic methods for drug discovery

Alex Dömling

11/03/2019

Press/Media: Research › Academic

Bedumer Winterloop 2016

Alex Dömling

06/02/2016

Press/Media: Public Engagement Activities › Popular

Zesde editie Bedumer Winterloop

Alex Dömling

28/01/2016

Press/Media: Public Engagement Activities › Popular

All (10) press/media

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