1. Rational Adaptation of L3MBTL1 Inhibitors to Create Small-Molecule Cbx7 Antagonists

   Simhadri, C., Daze, K. D., Douglas, S. F., Milosevich, N., Monjas, L., Dev, A., Brown, T. M., Hirsch, A. K. H., Wulff, J. E. & Hof, F., 6-Aug-2019, In : ChemMedChem. 14, 15, p. 1444-1456 13 p.

   Research output: Contribution to journal › Article › Academic › peer-review

2. Optimized Inhibitors of MDM2 via an Attempted Protein-Templated Reductive Amination

   van der Vlag, R., Unver, M. Y., Felicetti, T., Twarda-Clapa, A., Kassim, F., Ermis, C., Neochoritis, C. G., Musielak, B., Labuzek, B., Domling, A., Holak, T. A. & Hirsch, A. K. H., 12-Dec-2019, In : ChemMedChem. 14, 7 p.

   Research output: Contribution to journal › Article › Academic › peer-review

3. Anticancer Gold(III) Peptidomimetics: From Synthesis to in vitro and ex vivo Biological Evaluations

   Boscutti, G., Nardon, C., Marchio, L., Crisma, M., Biondi, B., Dalzoppo, D., Dalla Via, L., Formaggio, F., Casini, A. & Fregona, D., 6-Jun-2018, In : ChemMedChem. 13, 11, p. 1131-1145 15 p.

   Research output: Contribution to journal › Article › Academic › peer-review

4. Design and Synthesis of Bioisosteres of Acylhydrazones as Stable Inhibitors of the Aspartic Protease Endothiapepsin

   Jumde, V. R., Mondal, M., Gierse, R. M., Unver, M. Y., Magari, F., van Lier, R. C. W., Heine, A., Klebe, G. & Hirsch, A. K. H., 6-Nov-2018, In : ChemMedChem. 13, 21, p. 2266-2270 5 p.

   Research output: Contribution to journal › Article › Academic › peer-review

5. Anticancer Gold N-Heterocyclic Carbene Complexes: A Comparative in vitro and ex vivo Study

   Estrada-Ortiz, N., Guarra, F., de Graaf, I. A. M., Marchetti, L., de Jager, M. H., Groothuis, G. M. M., Gabbiani, C. & Casini, A., 7-Sep-2017, In : ChemMedChem. 12, 17, p. 1429-1435 7 p.

   Research output: Contribution to journal › Article › Academic › peer-review

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