1. The tale of proteolysis targeting chimeras (PROTACs) for leucine-rich repeat kinase 2 (LRRK2)

   Konstantinidou, M., Oun, A., Pathak, P., Zhang, B., Wang, Z., ter Brake, F., Dolga, A., Kortholt, A. & Doemling, A., 5-Dec-2020, In : ChemMedChem.

   Research output: Contribution to journal › Article › Academic › peer-review

2. Potential Dental Biofilm Inhibitors: Dynamic Combinatorial Chemistry Affords Sugar-Based Molecules that Target Bacterial Glucosyltransferase

   Hartman, A. M., Jumde, V. R., Elgaher, W. A. M., Te Poele, E. M., Dijkhuizen, L. & Hirsch, A. K. H., 8-Jan-2021, In : ChemMedChem. 16, 1, p. 113-123 11 p., cmdc.202000222.

   Research output: Contribution to journal › Article › Academic › peer-review

3. Rapid Discovery of Aspartyl Protease Inhibitors Using an Anchoring Approach

   Konstantinidou, M., Magari, F., Sutanto, F., Haupenthal, J., Jumde, V. R., Ünver, M. Y., Heine, A., Camacho, C. J., Hirsch, A. K. H., Klebe, G. & Dömling, A., 20-Apr-2020, In : ChemMedChem. 15, 8, p. 680-684 5 p.

   Research output: Contribution to journal › Article › Academic › peer-review

4. Rational Adaptation of L3MBTL1 Inhibitors to Create Small-Molecule Cbx7 Antagonists

   Simhadri, C., Daze, K. D., Douglas, S. F., Milosevich, N., Monjas, L., Dev, A., Brown, T. M., Hirsch, A. K. H., Wulff, J. E. & Hof, F., 6-Aug-2019, In : ChemMedChem. 14, 15, p. 1444-1456 13 p.

   Research output: Contribution to journal › Article › Academic › peer-review

5. Optimized Inhibitors of MDM2 via an Attempted Protein-Templated Reductive Amination

   van der Vlag, R., Unver, M. Y., Felicetti, T., Twarda-Clapa, A., Kassim, F., Ermis, C., Neochoritis, C. G., Musielak, B., Labuzek, B., Domling, A., Holak, T. A. & Hirsch, A. K. H., 17-Feb-2020, In : ChemMedChem. 15, 4, p. 370-375 7 p.

   Research output: Contribution to journal › Article › Academic › peer-review

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