1. Dynamic Combinatorial Chemistry Affords Sugar-Based Molecules Targeting Bacterial Glucosyltranseferase as Potential Dental Biofilm Inhibitors

   Hartman, A. M., Jumde, V. R., Elgaher, W. A. M., Te Poele, E. M., Dijkhuizen, L. & Hirsch, A. K. H., 16-Jun-2020, In : ChemMedChem. 11 p., cmdc.202000222.

   Research output: Contribution to journal › Article › Academic › peer-review

2. Rapid Discovery of Aspartyl Protease Inhibitors Using an Anchoring Approach

   Konstantinidou, M., Magari, F., Sutanto, F., Haupenthal, J., Jumde, V. R., Ünver, M. Y., Heine, A., Camacho, C. J., Hirsch, A. K. H., Klebe, G. & Dömling, A., 20-Apr-2020, In : ChemMedChem. 15, 8, p. 680-684 5 p.

   Research output: Contribution to journal › Article › Academic › peer-review

3. Rational Adaptation of L3MBTL1 Inhibitors to Create Small-Molecule Cbx7 Antagonists

   Simhadri, C., Daze, K. D., Douglas, S. F., Milosevich, N., Monjas, L., Dev, A., Brown, T. M., Hirsch, A. K. H., Wulff, J. E. & Hof, F., 6-Aug-2019, In : ChemMedChem. 14, 15, p. 1444-1456 13 p.

   Research output: Contribution to journal › Article › Academic › peer-review

4. Optimized Inhibitors of MDM2 via an Attempted Protein-Templated Reductive Amination

   van der Vlag, R., Unver, M. Y., Felicetti, T., Twarda-Clapa, A., Kassim, F., Ermis, C., Neochoritis, C. G., Musielak, B., Labuzek, B., Domling, A., Holak, T. A. & Hirsch, A. K. H., 17-Feb-2020, In : ChemMedChem. 15, 4, p. 370-375 7 p.

   Research output: Contribution to journal › Article › Academic › peer-review

5. Anticancer Gold(III) Peptidomimetics: From Synthesis to in vitro and ex vivo Biological Evaluations

   Boscutti, G., Nardon, C., Marchio, L., Crisma, M., Biondi, B., Dalzoppo, D., Dalla Via, L., Formaggio, F., Casini, A. & Fregona, D., 6-Jun-2018, In : ChemMedChem. 13, 11, p. 1131-1145 15 p.

   Research output: Contribution to journal › Article › Academic › peer-review

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