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Over ons Faculty of Science and Engineering Our Research GRIP Drug Design

Publications and Dissertations

Overview of publications of the research group Drug Design

Recent dissertations:

Click on the title to go to the pdf of the thesis:

Abdelraheem, E.M.M., Exploitation of macrocyclic chemical space by multicomponent reaction (MCR) and their applications in medicinal chemistry (2018)

Al-Qahtani, A., Production of novel protein therapeutics to improve targeted cancer therapy (2019)

Ali, A., Stapled peptides inhibitors: A new window for target drug discovery (2019)

Bashraheel, S., Studies on superantigens and antibody directed enzyme prodrug therapy for tolerable targeted cancer treatment (2019)

Batista, F.A. de, The oligomeric protein interference assay method for validation of antimalarial targets (2019)

Boltjes, A., Development and application of novel scaffolds in drug discovery: the MCR approach (2019)

Bosch, S.S., Analysis of the ATCase catalysis within the amino acid metabolism of the human malaria parasite Plasmodium falciparum (2019)

Gao, K., Structure-based drug discovery aiming at human-diseases related protein targets. (2020)

Gao, L., Multicomponent reactions in high throughput synthesis and medicinal chemistry (2022)

Gierse, R., Design, Synthesis and Structural Characterisation of Inhibitors of 1-Deoxy-D-xylulose-5-phosphate Synthase (2022)

Konstantinidou, M., Multicomponent reactions, applications in medicinal chemistry & new modalities in drug discovery (2020)

Li, J., Substrate exploitation of multicomponent reactions toward diverse scaffolds and applications in medicinal chemistry (2021)

Reyes Romero, A., Fragment-based Discovery Aiming at a Novel Modulation of Malate Dehydrogenase and Beyond (2021)

Ruiz Moreno, A.J., In Silico Design and Selection of CD44 Antagonists: implementation of computational methodologies in drug discovery and design (2021)

Sutanto, F., Development of Novel Covalent Inhibitors and Other Scaffolds Through Multicomponent Reactions (2020)

Wang, C., Allosteric inhibitors of aspartate transcarbamoylase: targeting pyrimidine biosynthesis to address multiple diseases (2023)

Wang, Q., MCR-based exploitation and application of diverse (poly)heterocyclic scaffolds (2020)

Wang, W., Applications of biophysical methods in small-molecule modulators targeting protein function (2020)

Wang, Z., Targeted protein degradation and multicomponent reactions in drug discovery (2022)

Xu, R., Diverse Substrate Scaffolds by Multicomponent Reactions and Protein Structural Dynamics by Single-molecule FRET (2022)

Laatst gewijzigd:23 juni 2023 08:52